لم تعد النسخة القابلة للطباعة مدعومة وقد تحتوي على أخطاء في العرض. يرجى تحديث علامات متصفحك المرجعية واستخدام وظيفة الطباعة الافتراضية في متصفحك بدلا منها.
تيميلاستين Temelastine هو مضاد هيستامين جديد مناهض انتقائي لمستقبلات H1. لا يعبر الجهاز العصبي المركزي.
الصيغة الكيميائية
C21H24BrN5O
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حسب المستقبل
Receptor | | Agonists: 2-Pyridylethylamine * Betahistine * Histamine * HTMT * UR-AK49Antagonists: 1st generation: 4-Methyldiphenhydramine * Alimemazine * Antazoline * Azatadine * Bamipine* Benzatropine/Benztropine * Bepotastine * Bromazine * Brompheniramine * Buclizine * Captodiame * Carbinoxamine * Chlorcyclizine * Chloropyramine * Chlorothen * Chlorphenamine * Chlorphenoxamine * Cinnarizine* Clemastine * Clobenzepam * Clocinizine * Cyclizine * Cyproheptadine * Dacemazine * Deptropine* Dexbrompheniramine * Dexchlorpheniramine * Dimenhydrinate * Dimetindene * Diphenhydramine * Diphenylpyraline * Doxylamine * Embramine * Etodroxizine * Etybenzatropine/Ethylbenztropine * Etymemazine * Flunarizine * Histapyrrodine * Homochlorcyclizine * Hydroxyethylpromethazine * Hydroxyzine * Isopromethazine * Isothipendyl * Meclozine * Mepyramine/Pyrilamine * Mequitazine * Methafurylene * Methapyrilene * Methdilazine * Moxastine * Niaprazine * Orphenadrine * Oxatomide * Oxomemazine * Phenindamine * Pheniramine * Phenyltoloxamine * Pimethixene * Piperoxan * Pipoxizine * Promethazine * Propiomazine * Pyrrobutamine * Talastine * Thenalidine * Thenyldiamine * Thiazinamium * Thonzylamine * Tolpropamine * Tripelennamine * Triprolidine
2nd generation: Acrivastine * Alinastine * Astemizole * Azelastine * Bamirastine * Barmastine * Bepiastine* Bepotastine * Bilastine * Cabastinen * Carebastine * Cetirizine * Clemastine * Clemizole * Clobenztropine * Dorastine * Ebastine * Emedastine * Epinastine * Flezelastine * Ketotifen * Latrepirdine* Levocabastine * Linetastine * Loratadine * Mapinastine * Mebhydrolin * Mizolastine * Moxastine * Noberastine * Octastine * Olopatadine * Perastine * Piclopastine * Rocastine * Rupatadine * Setastine * Talastine * Temelastine * Terfenadine * Zepastine
3rd generation: Desloratadine * Fexofenadine * Levocetirizine
Ungrouped: Belarizine * Efletirizine * Elbanizine * Flotrenizine * Medrylamine * Napactadine * Pibaxizine* Tagorizine * Trelnarizine * Trenizine * Vapitadine
Miscellaneous: Tricyclic antidepressants ( amitriptyline, * doxepin, * trimipramine, etc) * Tetracyclic antidepressants ( mianserin, * mirtazapine, etc) * Typical antipsychotics ( chlorpromazine, * thioridazine, etc) * Atypical antipsychotics ( clozapine, * olanzapine, * quetiapine, etc) |
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حسب الناقل العصبي
Transporter | |
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حسب الإنزيم
Enzyme | |
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