الفرق بين المراجعتين لصفحة: «قالب:هيستامينات»

من موسوعة العلوم العربية
اذهب إلى التنقل اذهب إلى البحث
(تحديث)
لا ملخص تعديل
 
(مراجعتان متوسطتان بواسطة مستخدم واحد آخر غير معروضتين)
سطر 1: سطر 1:
{{Navbox
{{Navbox
| name  = Histaminergics
| name  = الهيستامينات
| title = الهيستامينات<br />
| title = الهيستامينات<br />
(الناهضات والمثبطات)<br />
(الناهضات والمثبطات)<br />
سطر 16: سطر 16:
     | group1 = [[Histamine H1 receptor|H<sub>1</sub>]]
     | group1 = [[Histamine H1 receptor|H<sub>1</sub>]]
     |  list1 =
     |  list1 =
* '''Agonists''': [[2-Pyridylethylamine]]
'''Agonists''': [[2-Pyridylethylamine]] * [[Betahistine]] * [[Histamine]] * [[Histamine trifluoromethyl toluidide|HTMT]] * [[UR-AK49]]<br/>'''Antagonists''': ''1st generation'': [[4-Methyldiphenhydramine]] * [[Alimemazine]] * [[Antazoline]] * [[Azatadine]] * [[Bamipine]]*[[Benzatropine|Benzatropine/Benztropine]] * [[Bepotastine]] * [[Bromazine]] * [[Brompheniramine]] * [[Buclizine]] * [[Captodiame]] * [[Carbinoxamine]] * [[Chlorcyclizine]] * [[Chloropyramine]] * [[Chlorothen]] * [[Chlorphenamine]] * [[Chlorphenoxamine]] * [[Cinnarizine]]* [[Clemastine]] * [[Clobenzepam]] * [[Clocinizine]] * [[Cyclizine]] * [[Cyproheptadine]] * [[Dacemazine]] * [[Deptropine]]* [[Dexbrompheniramine]] * [[Dexchlorpheniramine]] * [[Dimenhydrinate]] * [[Dimetindene]] * [[Diphenhydramine]] * [[Diphenylpyraline]] * [[Doxylamine]] * [[Embramine]] * [[Etodroxizine]] * [[Etybenzatropine|Etybenzatropine/Ethylbenztropine]] * [[Etymemazine]] * [[Flunarizine]] * [[Histapyrrodine]] * [[Homochlorcyclizine]] * [[Hydroxyethylpromethazine]] * [[Hydroxyzine]] * [[Isopromethazine]] * [[Isothipendyl]] * [[Meclozine]] * [[Mepyramine|Mepyramine/Pyrilamine]] * [[Mequitazine]] * [[Methafurylene]] * [[Methapyrilene]] * [[Methdilazine]] * [[Moxastine]] * [[Niaprazine]] * [[Orphenadrine]] * [[Oxatomide]] * [[Oxomemazine]] * [[Phenindamine]] * [[Pheniramine]] * [[Phenyltoloxamine]] * [[Pimethixene]] * [[Piperoxan]] * [[Pipoxizine]] * [[Promethazine]] * [[Propiomazine]] * [[Pyrrobutamine]] * [[Talastine]] * [[Thenalidine]] * [[Thenyldiamine]] * [[Thiazinamium]] * [[Thonzylamine]] * [[Tolpropamine]] * [[Tripelennamine]] * [[Triprolidine]]
* [[Betahistine]]
* [[Histamine]]
* [[Histamine trifluoromethyl toluidide|HTMT]]
* [[UR-AK49]]<br/>'''Antagonists''': ''1st generation'': [[4-Methyldiphenhydramine]]
* [[Alimemazine]]
* [[Antazoline]]
* [[Azatadine]]
* [[Bamipine]]
* [[Benzatropine|Benzatropine/Benztropine]]
* [[Bepotastine]]
* [[Bromazine]]
* [[Brompheniramine]]
* [[Buclizine]]
* [[Captodiame]]
* [[Carbinoxamine]]
* [[Chlorcyclizine]]
* [[Chloropyramine]]
* [[Chlorothen]]
* [[Chlorphenamine]]
* [[Chlorphenoxamine]]
* [[Cinnarizine]]
* [[Clemastine]]
* [[Clobenzepam]]
* [[Clocinizine]]
* [[Cyclizine]]
* [[Cyproheptadine]]
* [[Dacemazine]]
* [[Deptropine]]
* [[Dexbrompheniramine]]
* [[Dexchlorpheniramine]]
* [[Dimenhydrinate]]
* [[Dimetindene]]
* [[Diphenhydramine]]
* [[Diphenylpyraline]]
* [[Doxylamine]]
* [[Embramine]]
* [[Etodroxizine]]
* [[Etybenzatropine|Etybenzatropine/Ethylbenztropine]]
* [[Etymemazine]]
* [[Flunarizine]]
* [[Histapyrrodine]]
* [[Homochlorcyclizine]]
* [[Hydroxyethylpromethazine]]
* [[Hydroxyzine]]
* [[Isopromethazine]]
* [[Isothipendyl]]
* [[Meclozine]]
* [[Mepyramine|Mepyramine/Pyrilamine]]
* [[Mequitazine]]
* [[Methafurylene]]
* [[Methapyrilene]]
* [[Methdilazine]]
* [[Moxastine]]
* [[Niaprazine]]
* [[Orphenadrine]]
* [[Oxatomide]]
* [[Oxomemazine]]
* [[Phenindamine]]
* [[Pheniramine]]
* [[Phenyltoloxamine]]
* [[Pimethixene]]
* [[Piperoxan]]
* [[Pipoxizine]]
* [[Promethazine]]
* [[Propiomazine]]
* [[Pyrrobutamine]]
* [[Talastine]]
* [[Thenalidine]]
* [[Thenyldiamine]]
* [[Thiazinamium]]
* [[Thonzylamine]]
* [[Tolpropamine]]
* [[Tripelennamine]]
* [[Triprolidine]]


* ''2nd generation'': [[Acrivastine]]
''2nd generation'': [[Acrivastine]] * [[Alinastine]] * [[Astemizole]] * [[Azelastine]] * [[Bamirastine]] * [[Barmastine]] * [[Bepiastine]]* [[Bepotastine]] * [[Bilastine]] * [[Cabastinen]] * [[Carebastine]] * [[Cetirizine]] * [[Clemastine]] * [[Clemizole]] * [[Clobenztropine]] * [[Dorastine]] * [[Ebastine]] * [[Emedastine]] * [[Epinastine]] * [[Flezelastine]] * [[Ketotifen]] * [[Latrepirdine]]* [[Levocabastine]] * [[Linetastine]] * [[Loratadine]] * [[Mapinastine]] * [[Mebhydrolin]] * [[Mizolastine]] * [[Moxastine]] * [[Noberastine]] * [[Octastine]] * [[Olopatadine]] * [[Perastine]] * [[Piclopastine]] * [[Rocastine]] * [[Rupatadine]] * [[Setastine]] * [[Talastine]] * [[Temelastine]] * [[Terfenadine]] * [[Zepastine]]
* [[Alinastine]]
* [[Astemizole]]
* [[Azelastine]]
* [[Bamirastine]]
* [[Barmastine]]
* [[Bepiastine]]
* [[Bepotastine]]
* [[Bilastine]]
* [[Cabastinen]]
* [[Carebastine]]
* [[Cetirizine]]
* [[Clemastine]]
* [[Clemizole]]
* [[Clobenztropine]]
* [[Dorastine]]
* [[Ebastine]]
* [[Emedastine]]
* [[Epinastine]]
* [[Flezelastine]]
* [[Ketotifen]]
* [[Latrepirdine]]
* [[Levocabastine]]
* [[Linetastine]]
* [[Loratadine]]
* [[Mapinastine]]
* [[Mebhydrolin]]
* [[Mizolastine]]
* [[Moxastine]]
* [[Noberastine]]
* [[Octastine]]
* [[Olopatadine]]
* [[Perastine]]
* [[Piclopastine]]
* [[Rocastine]]
* [[Rupatadine]]
* [[Setastine]]
* [[Talastine]]
* [[Temelastine]]
* [[Terfenadine]]
* [[Zepastine]]


* ''3rd generation'': [[Desloratadine]]
''3rd generation'': [[Desloratadine]] * [[Fexofenadine]] * [[Levocetirizine]]
* [[Fexofenadine]]
* [[Levocetirizine]]


* ''Ungrouped'': [[Belarizine]]
''Ungrouped'': [[Belarizine]] * [[Efletirizine]] * [[Elbanizine]] * [[Flotrenizine]] * [[Medrylamine]] * [[Napactadine]] * [[Pibaxizine]]* [[Tagorizine]] * [[Trelnarizine]] * [[Trenizine]] * [[Vapitadine]]
* [[Efletirizine]]
* [[Elbanizine]]
* [[Flotrenizine]]
* [[Medrylamine]]
* [[Napactadine]]
* [[Pibaxizine]]
* [[Tagorizine]]
* [[Trelnarizine]]
* [[Trenizine]]
* [[Vapitadine]]


* ''Miscellaneous'': [[Tricyclic antidepressant]]s ([[amitriptyline]],  
''Miscellaneous'': [[Tricyclic antidepressant]]s ([[amitriptyline]], * [[doxepin]], * [[trimipramine]], etc) * [[Tetracyclic antidepressant]]s ([[mianserin]], * [[mirtazapine]], etc) * [[Typical antipsychotic]]s ([[chlorpromazine]], * [[thioridazine]], etc) * [[Atypical antipsychotic]]s ([[clozapine]], * [[olanzapine]], * [[quetiapine]], etc)
* [[doxepin]],  
* [[trimipramine]], etc)
* [[Tetracyclic antidepressant]]s ([[mianserin]],  
* [[mirtazapine]], etc)
* [[Typical antipsychotic]]s ([[chlorpromazine]],  
* [[thioridazine]], etc)
* [[Atypical antipsychotic]]s ([[clozapine]],  
* [[olanzapine]],  
* [[quetiapine]], etc)


     | group2 = [[Histamine H2 receptor|H<sub>2</sub>]]
     | group2 = [[Histamine H2 receptor|H<sub>2</sub>]]
     |  list2 =
     |  list2 =
* '''Agonists''': [[Amthamine]]
'''Agonists''': [[Amthamine]] * [[Betazole]] * [[Dimaprit]] * [[Histamine]] * [[Histamine trifluoromethyl toluidide|HTMT]] * [[Impromidine]] * [[UR-AK49]]<br/>'''Antagonists''': [[Bisfentidine]] [[Burimamide]] * [[Cimetidine]] * [[Dalcotidine]] * [[Donetidine]] * [[Ebrotidine]] * [[Etintidine]] * [[Famotidine]] * [[Lafutidine]] * [[Lamtidine]] * [[Lavoltidine|Lavoltidine/Loxtidine]] * [[Lupitidine]] * [[Metiamide]]* [[Mifentidine]] * [[Niperotidine]] * [[Nizatidine]] * [[Osutidine]] * [[Oxmetidine]] * [[Pibutidine]] * [[Quisultazine|Quisultazine/Quisultidine]] * [[Ramixotidine]] * [[Ranitidine]] * [[Roxatidine]] * [[Sufotidine]] * [[Tiotidine]] * [[Tuvatidine]] * [[Venritidine]] * [[Xaltidine]]
* [[Betazole]]
* [[Dimaprit]]
* [[Histamine]]
* [[Histamine trifluoromethyl toluidide|HTMT]]
* [[Impromidine]]
* [[UR-AK49]]<br/>'''Antagonists''': [[Bisfentidine]]
* [[Burimamide]]
* [[Cimetidine]]
* [[Dalcotidine]]
* [[Donetidine]]
* [[Ebrotidine]]
* [[Etintidine]]
* [[Famotidine]]
* [[Lafutidine]]
* [[Lamtidine]]
* [[Lavoltidine|Lavoltidine/Loxtidine]]
* [[Lupitidine]]
* [[Metiamide]]
* [[Mifentidine]]
* [[Niperotidine]]
* [[Nizatidine]]
* [[Osutidine]]
* [[Oxmetidine]]
* [[Pibutidine]]
* [[Quisultazine|Quisultazine/Quisultidine]]
* [[Ramixotidine]]
* [[Ranitidine]]
* [[Roxatidine]]
* [[Sufotidine]]
* [[Tiotidine]]
* [[Tuvatidine]]
* [[Venritidine]]
* [[Xaltidine]]


     | group3 = [[Histamine H3 receptor|H<sub>3</sub>]]
     | group3 = [[Histamine H3 receptor|H<sub>3</sub>]]
     |  list3 =
     |  list3 =
* '''Agonists''': [[alpha-Methylhistamine|ل-Methylhistamine]]
'''Agonists''': [[alpha-Methylhistamine|ل-Methylhistamine]] * [[Cipralisant]] * [[Histamine]] * [[Imetit]] * [[Immepip]] * [[Immethridine]] * [[Methimepip]] * [[Proxyfan]]<br/>'''Antagonists''': [[A-349,821]] * [[A-423,579]] * [[ABT-239]] * [[Betahistine]] * [[Burimamide]] * [[Ciproxifan]] * [[Clobenpropit]] * [[Conessine]] * [[GSK-189,254]] * [[Impentamine]] * [[Iodophenpropit]] * [[JNJ-5207852|JNJ-5,207,852]] * [[MK-0249]] * [[NNC 38-1049|NNC-38-1,049]] * [[PF-03654746]] * [[Pitolisant]] * [[SCH-79687|SCH-79,687]] * [[Thioperamide]] * [[VUF-5681|VUF-5,681]]
* [[Cipralisant]]
* [[Histamine]]
* [[Imetit]]
* [[Immepip]]
* [[Immethridine]]
* [[Methimepip]]
* [[Proxyfan]]<br/>'''Antagonists''': [[A-349,821]]
* [[A-423,579]]
* [[ABT-239]]
* [[Betahistine]]
* [[Burimamide]]
* [[Ciproxifan]]
* [[Clobenpropit]]
* [[Conessine]]
* [[GSK-189,254]]
* [[Impentamine]]
* [[Iodophenpropit]]
* [[JNJ-5207852|JNJ-5,207,852]]
* [[MK-0249]]
* [[NNC 38-1049|NNC-38-1,049]]
* [[PF-03654746]]
* [[Pitolisant]]
* [[SCH-79687|SCH-79,687]]
* [[Thioperamide]]
* [[VUF-5681|VUF-5,681]]


     | group4 = [[Histamine H4 receptor|H<sub>4</sub>]]
     | group4 = [[Histamine H4 receptor|H<sub>4</sub>]]
     |  list4 =
     |  list4 =
* '''Agonists''': [[4-Methylhistamine]]
'''Agonists''': [[4-Methylhistamine]] * [[Histamine]] * [[VUF-8430|VUF-8,430]]<br/>'''Antagonists''': [[JNJ-7777120|JNJ-7,777,120]] [[Thioperamide]] * [[VUF-6002|VUF-6,002]]
* [[Histamine]]
* [[VUF-8430|VUF-8,430]]<br/>'''Antagonists''': [[JNJ-7777120|JNJ-7,777,120]]
* [[Thioperamide]]
* [[VUF-6002|VUF-6,002]]


   }}
   }}
سطر 244: سطر 47:
     | group1 = [[Vesicular monoamine transporter|VMAT]]
     | group1 = [[Vesicular monoamine transporter|VMAT]]
     | list1  =
     | list1  =
* '''Inhibitors:''' [[Ibogaine]]
'''Inhibitors:''' [[Ibogaine]] * [[Reserpine]] * [[Tetrabenazine]]
* [[Reserpine]]
* [[Tetrabenazine]]


   }}
   }}
سطر 257: سطر 58:
     | group1 = [[Histidine decarboxylase|HDC]]
     | group1 = [[Histidine decarboxylase|HDC]]
     | list1  =
     | list1  =
* '''Inhibitors:''' [[(+)-Catechin|Catechin]]
'''Inhibitors:''' [[(+)-Catechin|Catechin]] * [[Meciadanol]] * [[Naringenin]] * [[Tritoqualine]]
* [[Meciadanol]]
* [[Naringenin]]
* [[Tritoqualine]]


     | group2 = [[Histamine N-methyltransferase|HNMT]]
     | group2 = [[Histamine N-methyltransferase|HNMT]]
     | list2  =
     | list2  =
* '''Inhibitors:''' [[Amodiaquine]]
'''Inhibitors:''' [[Amodiaquine]] * [[Diphenhydramine]] * [[Harmaline]] * [[Metoprine]] * [[Quinacrine]] * [[SKF-91,488]] * [[Tacrine]]
* [[Diphenhydramine]]
* [[Harmaline]]
* [[Metoprine]]
* [[Quinacrine]]
* [[SKF-91,488]]
* [[Tacrine]]


     | group2 = [[Diamine oxidase|DAO]]
     | group2 = [[Diamine oxidase|DAO]]
     | list2  =
     | list2  =
* '''Inhibitors:''' [[Aminoguanidine]]
'''Inhibitors:''' [[Aminoguanidine]]


   }}
   }}
سطر 284: سطر 76:
     | group1 = Endogenous
     | group1 = Endogenous
     | list1  =
     | list1  =
* [[Histamine]]; ''Precursors:'' [[L-Histidine|<small>L</small>-Histidine]]; ''Cofactors:'' [[Vitamin B6]]
[[Histamine]]; ''Precursors:'' [[L-Histidine|<small>L</small>-Histidine]]; ''Cofactors:'' [[Vitamin B6]]


   }}
   }}

المراجعة الحالية بتاريخ 18:12، 18 يناير 2013